A Chemical-Biological Study Reveals C-9-type Iridoids as Novel Heat Shock Protein 90 (Hsp90) Inhibitors
2013-01-01 Dal Piaz, F.; Vassallo, A.; Temraz, A.; Cotugno, R.; Belisario, M. A .; Bifulco, G.; Chini, M. G.; Pisano, C.; De Tommasi, N.; Braca, A.
The Binding Mode of Cladocoran A to the Human Group IIA Phospholipase A2
2011-01-01 Monti, M. C.; Chini, M. G.; Margarucci, L.; Riccio, R.; Bifulco, G.; Casapullo, A.
Preliminary Structure-Activity Relationship on Theonellasterol, a New Chemotype of FXR Antagonist, from the Marine Sponge Theonella swinhoei
2012-01-01 Sepe, Valentina; Ummarino, Raffaella; D'Auria, Maria; Taglialatela-Scafati, Orazio; Marino, Simona; D'Amore, Claudio; Renga, Barbara; Chini, Maria Giovanna; Bifulco, Giuseppe; Nakao, Yoichi; Fusetani, Nobuhiro; Fiorucci, Stefano; Zampella, Angela
Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors
2016-01-01 Terracciano, Stefania; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Targeting the Hsp90 C-terminal domain by the chemically accessible dihydropyrimidinone scaffold
2015-01-01 Strocchia, Maria; Terracciano, Stefania; Chini, MARIA GIOVANNA; Vassallo, Antonio; Vaccaro, Maria C.; DAL PIAZ, Fabrizio; Leone, Antonietta; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
New dihydropyrimidin-2(1H)-one based Hsp90 C-terminal inhibitors
2016-01-01 Terracciano, Stefania; Foglia, Antonio; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Russo, Alessandra; DAL PIAZ, Fabrizio; Saturnino, C.; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Conformationally locked calixarene-based histone deacetylase inhibitors
2010-01-01 Chini, M. G.; Terracciano, S.; Riccio, R.; Bifulco, G.; Ciao, R.; Gaeta, C.; Troisi, F.; Neri, P.
Synthesis, Biological Evaluation, and Molecular Docking of Ugi Products Containing a Zinc-Chelating Moiety as Novel Inhibitors of Histone Deacetylases
2009-01-01 Grolla, Aa; Podesta, V; Chini, M. G.; DI MICCO, S; Vallario, A; Genazzani, Aa; Canonico, Pl; Bifulco, G; Tron, Gc; Sorba, G; Pirali, T
Correction: Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors
2016-01-01 Terracciano, Stefania; Chini, Maria Giovanna; Vaccaro, Mariacarmela; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Conicasterol E, a Small Heterodimer Partner Sparing Farnesoid X Receptor Modulator Endowed with a Pregnane X Receptor Agonistic Activity, from the Marine SpongeTheonella swinhoei
2012-01-01 Sepe, Valentina; Ummarino, Raffaella; Valeria D’Auria, Maria; Chini, Maria Giovanna; Bifulco, Giuseppe; Renga, Barbara; D’Amore, Claudio; Debitus, Cécile; Fiorucci, Stefano; Zampella, Angela
The Inactivation Mechanism of Human Group IIA Phospholipase A2by Scalaradial
2012-01-01 Margarucci, Luigi; Monti, Maria Chiara; Chini, MARIA GIOVANNA; Tosco, Alessandra; Riccio, Raffaele; Bifulco, Giuseppe; Casapullo, Agostino
The molecular mechanism of human group IIA phospholipase A2 inactivation by bolinaquinone
2009-01-01 Monti, Maria Chiara; Chini, MARIA GIOVANNA; Margarucci, Luigi; Tosco, Alessandra; Riccio, Raffaele; Bifulco, Giuseppe; Casapullo, Agostino
Design, Synthesis, and Biological Activity of Hydroxamic Tertiary Amines as Histone Deacetylase Inhibitors
2012-01-01 Terracciano, Stefania; Chini, Maria Giovanna; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
4-Methylenesterols from Theonella swinhoei sponge are natural pregnane-X-receptor agonists and farnesoid-X-receptor antagonists that modulate innate immunity
2012-01-01 De Marino, Simona; Ummarino, Raffaella; Valeria D’Auria, Maria; Chini, Maria Giovanna; Bifulco, Giuseppe; D’Amore, Claudio; Renga, Barbara; Mencarelli, Andrea; Petek, Sylvain; Fiorucci, Stefano; Zampella, Angela
Use of NMR in profiling of cocaine seizures
2013-01-01 Bruno, Pagano; Ilaria, Lauri; Stefano De, Tito; Guido, Persico; Chini, M. G.; Anders, Malmendal; Ettore, Novellino; Antonio, Randazzo
Dimeric and trimeric triazole based molecules as a new class of Hsp90 molecular chaperone inhibitors
2013-01-01 Terracciano, Stefania; Chini, MARIA GIOVANNA; DAL PIAZ, Fabrizio; Antonio, Vassallo; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
Can Robots Save Us from Reification? New Responsibilities for a New Capitalism
2020-01-01 Abbate, Fabrizia
Haute cuisine and country of origin
2019-01-01 Presenza, A.; Messeni Petruzzelli, A.
Antagonistic Activity against Ascosphaera apis and Functional Properties of Lactobacillus kunkeei Strains
2020-01-01 Iorizzo, Massimo; Lombardi, Silvia Jane; Ganassi, Sonia; Testa, Bruno; Ianiro, Mario; Letizia, Francesco; Succi, Mariantonietta; Tremonte, Patrizio; Vergalito, Franca; Cozzolino, Autilia; Sorrentino, Elena; Coppola, Raffaele; Petrarca, Sonia; Mancini, Massimo; Cristofaro, Antonio De
Debunking Fake Humanities. Critical reasoning from Ovid to Roboethics
2019-01-01 Abbate, Fabrizia
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| A Chemical-Biological Study Reveals C-9-type Iridoids as Novel Heat Shock Protein 90 (Hsp90) Inhibitors | 1-gen-2013 | Dal Piaz, F.; Vassallo, A.; Temraz, A.; Cotugno, R.; Belisario, M. A .; Bifulco, G.; Chini, M. G.; Pisano, C.; De Tommasi, N.; Braca, A. | |
| The Binding Mode of Cladocoran A to the Human Group IIA Phospholipase A2 | 1-gen-2011 | Monti, M. C.; Chini, M. G.; Margarucci, L.; Riccio, R.; Bifulco, G.; Casapullo, A. | |
| Preliminary Structure-Activity Relationship on Theonellasterol, a New Chemotype of FXR Antagonist, from the Marine Sponge Theonella swinhoei | 1-gen-2012 | Sepe, Valentina; Ummarino, Raffaella; D'Auria, Maria; Taglialatela-Scafati, Orazio; Marino, Simona; D'Amore, Claudio; Renga, Barbara; Chini, Maria Giovanna; Bifulco, Giuseppe; Nakao, Yoichi; Fusetani, Nobuhiro; Fiorucci, Stefano; Zampella, Angela | |
| Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors | 1-gen-2016 | Terracciano, Stefania; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Targeting the Hsp90 C-terminal domain by the chemically accessible dihydropyrimidinone scaffold | 1-gen-2015 | Strocchia, Maria; Terracciano, Stefania; Chini, MARIA GIOVANNA; Vassallo, Antonio; Vaccaro, Maria C.; DAL PIAZ, Fabrizio; Leone, Antonietta; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| New dihydropyrimidin-2(1H)-one based Hsp90 C-terminal inhibitors | 1-gen-2016 | Terracciano, Stefania; Foglia, Antonio; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Russo, Alessandra; DAL PIAZ, Fabrizio; Saturnino, C.; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Conformationally locked calixarene-based histone deacetylase inhibitors | 1-gen-2010 | Chini, M. G.; Terracciano, S.; Riccio, R.; Bifulco, G.; Ciao, R.; Gaeta, C.; Troisi, F.; Neri, P. | |
| Synthesis, Biological Evaluation, and Molecular Docking of Ugi Products Containing a Zinc-Chelating Moiety as Novel Inhibitors of Histone Deacetylases | 1-gen-2009 | Grolla, Aa; Podesta, V; Chini, M. G.; DI MICCO, S; Vallario, A; Genazzani, Aa; Canonico, Pl; Bifulco, G; Tron, Gc; Sorba, G; Pirali, T | |
| Correction: Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors | 1-gen-2016 | Terracciano, Stefania; Chini, Maria Giovanna; Vaccaro, Mariacarmela; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Conicasterol E, a Small Heterodimer Partner Sparing Farnesoid X Receptor Modulator Endowed with a Pregnane X Receptor Agonistic Activity, from the Marine SpongeTheonella swinhoei | 1-gen-2012 | Sepe, Valentina; Ummarino, Raffaella; Valeria D’Auria, Maria; Chini, Maria Giovanna; Bifulco, Giuseppe; Renga, Barbara; D’Amore, Claudio; Debitus, Cécile; Fiorucci, Stefano; Zampella, Angela | |
| The Inactivation Mechanism of Human Group IIA Phospholipase A2by Scalaradial | 1-gen-2012 | Margarucci, Luigi; Monti, Maria Chiara; Chini, MARIA GIOVANNA; Tosco, Alessandra; Riccio, Raffaele; Bifulco, Giuseppe; Casapullo, Agostino | |
| The molecular mechanism of human group IIA phospholipase A2 inactivation by bolinaquinone | 1-gen-2009 | Monti, Maria Chiara; Chini, MARIA GIOVANNA; Margarucci, Luigi; Tosco, Alessandra; Riccio, Raffaele; Bifulco, Giuseppe; Casapullo, Agostino | |
| Design, Synthesis, and Biological Activity of Hydroxamic Tertiary Amines as Histone Deacetylase Inhibitors | 1-gen-2012 | Terracciano, Stefania; Chini, Maria Giovanna; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| 4-Methylenesterols from Theonella swinhoei sponge are natural pregnane-X-receptor agonists and farnesoid-X-receptor antagonists that modulate innate immunity | 1-gen-2012 | De Marino, Simona; Ummarino, Raffaella; Valeria D’Auria, Maria; Chini, Maria Giovanna; Bifulco, Giuseppe; D’Amore, Claudio; Renga, Barbara; Mencarelli, Andrea; Petek, Sylvain; Fiorucci, Stefano; Zampella, Angela | |
| Use of NMR in profiling of cocaine seizures | 1-gen-2013 | Bruno, Pagano; Ilaria, Lauri; Stefano De, Tito; Guido, Persico; Chini, M. G.; Anders, Malmendal; Ettore, Novellino; Antonio, Randazzo | |
| Dimeric and trimeric triazole based molecules as a new class of Hsp90 molecular chaperone inhibitors | 1-gen-2013 | Terracciano, Stefania; Chini, MARIA GIOVANNA; DAL PIAZ, Fabrizio; Antonio, Vassallo; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| Can Robots Save Us from Reification? New Responsibilities for a New Capitalism | 1-gen-2020 | Abbate, Fabrizia | |
| Haute cuisine and country of origin | 1-gen-2019 | Presenza, A.; Messeni Petruzzelli, A. | |
| Antagonistic Activity against Ascosphaera apis and Functional Properties of Lactobacillus kunkeei Strains | 1-gen-2020 | Iorizzo, Massimo; Lombardi, Silvia Jane; Ganassi, Sonia; Testa, Bruno; Ianiro, Mario; Letizia, Francesco; Succi, Mariantonietta; Tremonte, Patrizio; Vergalito, Franca; Cozzolino, Autilia; Sorrentino, Elena; Coppola, Raffaele; Petrarca, Sonia; Mancini, Massimo; Cristofaro, Antonio De | |
| Debunking Fake Humanities. Critical reasoning from Ovid to Roboethics | 1-gen-2019 | Abbate, Fabrizia |
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