Synthesis of new mono and bis amides projected as potential histone deacetylase (HDAC) inhibitors
2010-01-01 Terracciano, Stefania; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; E., Damico; Marzocco, Stefania; Riccio, Raffaele; Bruno, Ines
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach
2016-01-01 Chini Maria, G.; Malafronte, Nicola; Vaccaro Maria, C.; Gualtieri Maria, J.; Vassallo, Antonio; Vasaturo, Michele; Castellano, Sabrina; Milite, Ciro; Leone, Antonietta; Bifulco, Giuseppe; De Tommasi, Nunziatina; Dal Piaz, Fabrizio
Can Small Chemical Modifications of Natural Pan-inhibitors Modulate the Biological Selectivity? the Case of Curcumin Prenylated Derivatives Acting as HDAC or mPGES-1 Inhibitors
2015-01-01 Iranshahi, Mehrdad; Chini, MARIA GIOVANNA; Masullo, Milena; Sahebkar, Amirhossein; Javidnia, Azita; Chitsazian Yazdi, Mahsa; Pergola, Carlo; Koeberle, Andreas; Werz, Oliver; Pizza, Cosimo; Terracciano, Stefania; Piacente, Sonia; Bifulco, Giuseppe
Guaianolides from Ormenis mixta: Structural Insights and Evaluation of Their Anti-inflammatory Profile
2019-01-01 Benteldjoune, Mounira; Chini, Maria Giovanna; Iannuzzi, Anna Maria; Kabouche, Ahmed; Kabouche, Zahia; Dʼambola, Massimiliano; Marzocco, Stefania; Autore, Giuseppina; Bifulco, Giuseppe; De Tommasi, Nunziatina
Quantum Mechanical Calculation of NMR Parameters in the Stereostructural Determination of Natural Products
2010-01-01 DI MICCO, Simone; Chini, MARIA GIOVANNA; Riccio, Raffaele; Bifulco, Giuseppe
Quantitative NMR-Derived Interproton Distances Combined with Quantum Mechanical Calculations of13C Chemical Shifts in the Stereochemical Determination of Conicasterol F, a Nuclear Receptor Ligand fromTheonella swinhoei
2012-01-01 Chini, Maria Giovanna; Jones, Catharine R.; Zampella, Angela; Valeria D’Auria, Maria; Renga, Barbara; Fiorucci, Stefano; Butts, Craig P.; Bifulco, Giuseppe
Identification and mechanism of action analysis of the new PARP-1 inhibitor 2″-hydroxygenkwanol A
2015-01-01 Dal Piaz, Fabrizio; Ferro, Piera; Vassallo, Antonio; Vasaturo, Michele; Forte, Giovanni; Chini, Maria Giovanna; Bifulco, Giuseppe; Tosco, Alessandra; De Tommasi, Nunziatina
Natural iminosugar (+)-lentiginosine inhibits ATPase and chaperone activity of Hsp90
2012-01-01 Dal Piaz, Fabrizio; Vassallo, Antonio; Chini, Maria Giovanna; Cordero Franca, M.; Cardona, Francesca; Pisano, Claudio; Bifulco, Giuseppe; De Tommasi, Nunziatina; Brandi, Alberto
Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells
2018-01-01 Khalfaoui, Ayoub; Chini, Maria G.; Bouheroum, Mohamed; Belaabed, Soumia; Lauro, Gianluigi; Terracciano, Stefania; Carmela Vaccaro, Maria; Bruno, Ines; Benayache, Samir; Mancini, Ines; Bifulco, Giuseppe
Molecular mechanism of tanshinone IIA and cryptotanshinone in platelet anti-aggregating effects: an integrated study of pharmacology and computational analysis
2015-01-01 Maione, Francesco; Cantone, Vincenza; Chini, MARIA GIOVANNA; DE FEO, Vincenzo; Mascolo, Nicola; Bifulco, Giuseppe
Structure-Based Discovery of Inhibitors of Microsomal Prostaglandin E2 Synthase-1, 5-Lipoxygenase and 5-Lipoxygenase-Activating Protein: Promising Hits for the Development of New Anti-inflammatory Agents
2011-01-01 De Simone, R.; Chini, M. G.; Bruno, I.; Riccio, R.; Mueller, D.; Werz, O.; Bifulco, G.
Fusicoccane Diterpenes from Hypoestes forsskaolii as Heat Shock Protein 90 (Hsp90) Modulators
2019-01-01 D'Ambola, Massimiliano; Fiengo, Lorenzo; Chini, Maria Giovanna; Cotugno, Roberta; Bader, Ammar; Bifulco, Giuseppe; Braca, Alessandra; De Tommasi, Nunziatina; Dal Piaz, Fabrizio
Discovery of new molecular entities able to strongly interfere with Hsp90 C-terminal domain
2018-01-01 Terracciano, Stefania; Russo, Alessandra; Chini, Maria G.; Vaccaro, Maria C.; Potenza, Marianna; Vassallo, Antonio; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
The bile acid receptor GPBAR-1 (TGR5) modulates integrity of intestinal barrier and immune response to experimental Colitis
2011-01-01 Cipriani, S.; Mencarelli, A.; Chini, M. G.; Distrutti, E.; Renga, B.; Bifulco, G.; Baldelli, F.; Donini, A.; Fiorucci, S.
Elucidating new structural features of the triazole scaffold for the development of mPGES-1 inhibitors
2015-01-01 Chini, MARIA GIOVANNA; Ferroni, Claudia; Cantone, Vincenza; Dambruoso, Paolo; Varchi, Greta; Pepe, Antonella; Fischer, Katrin; Pergola, Carlo; Werz, Oliver; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe
Computational NMR Methods in the Stereochemical Analysis of Organic Compounds: Are Proton or Carbon NMR Chemical Shift Data More Discriminating?
2015-01-01 Chini, MARIA GIOVANNA; Riccio, Raffaele; Bifulco, Giuseppe
Structural basis for the design and synthesis of selective HDAC inhibitors
2013-01-01 DI MICCO, Simone; Chini, MARIA GIOVANNA; Terracciano, Stefania; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe
Discovery That Theonellasterol a Marine Sponge Sterol Is a Highly Selective FXR Antagonist That Protects against Liver Injury in Cholestasis
2012-01-01 Barbara, Renga; Andrea, Mencarelli; Claudio, D'Amore; Sabrina, Cipriani; Maria Valeria, D'Auria; Valentina, Sepe; Chini, MARIA GIOVANNA; Monti, Maria Chiara; Bifulco, Giuseppe; Angela, Zampella; Stefano, Fiorucci
Design and synthesis of a second series of triazole-based compounds as potent dual mPGES-1 and 5-lipoxygenase inhibitors
2012-01-01 Chini, Maria Giovanna; De Simone, Rosa; Bruno, Ines; Riccio, Raffaele; Dehm, Friederike; Weinigel, Christina; Barz, Dagmar; Werz, Oliver; Bifulco, Giuseppe
A Novel Potent Nicotinamide Phosphoribosyltransferase Inhibitor Synthesized via Click Chemistry
2010-01-01 G., Colombano; C., Travelli; U., Galli; A., Caldarelli; Chini, MARIA GIOVANNA; P. L., Canonico; G., Sorba; Bifulco, Giuseppe; G. C., Tron; A. A., Genazzani
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Synthesis of new mono and bis amides projected as potential histone deacetylase (HDAC) inhibitors | 1-gen-2010 | Terracciano, Stefania; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; E., Damico; Marzocco, Stefania; Riccio, Raffaele; Bruno, Ines | |
| Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach | 1-gen-2016 | Chini Maria, G.; Malafronte, Nicola; Vaccaro Maria, C.; Gualtieri Maria, J.; Vassallo, Antonio; Vasaturo, Michele; Castellano, Sabrina; Milite, Ciro; Leone, Antonietta; Bifulco, Giuseppe; De Tommasi, Nunziatina; Dal Piaz, Fabrizio | |
| Can Small Chemical Modifications of Natural Pan-inhibitors Modulate the Biological Selectivity? the Case of Curcumin Prenylated Derivatives Acting as HDAC or mPGES-1 Inhibitors | 1-gen-2015 | Iranshahi, Mehrdad; Chini, MARIA GIOVANNA; Masullo, Milena; Sahebkar, Amirhossein; Javidnia, Azita; Chitsazian Yazdi, Mahsa; Pergola, Carlo; Koeberle, Andreas; Werz, Oliver; Pizza, Cosimo; Terracciano, Stefania; Piacente, Sonia; Bifulco, Giuseppe | |
| Guaianolides from Ormenis mixta: Structural Insights and Evaluation of Their Anti-inflammatory Profile | 1-gen-2019 | Benteldjoune, Mounira; Chini, Maria Giovanna; Iannuzzi, Anna Maria; Kabouche, Ahmed; Kabouche, Zahia; Dʼambola, Massimiliano; Marzocco, Stefania; Autore, Giuseppina; Bifulco, Giuseppe; De Tommasi, Nunziatina | |
| Quantum Mechanical Calculation of NMR Parameters in the Stereostructural Determination of Natural Products | 1-gen-2010 | DI MICCO, Simone; Chini, MARIA GIOVANNA; Riccio, Raffaele; Bifulco, Giuseppe | |
| Quantitative NMR-Derived Interproton Distances Combined with Quantum Mechanical Calculations of13C Chemical Shifts in the Stereochemical Determination of Conicasterol F, a Nuclear Receptor Ligand fromTheonella swinhoei | 1-gen-2012 | Chini, Maria Giovanna; Jones, Catharine R.; Zampella, Angela; Valeria D’Auria, Maria; Renga, Barbara; Fiorucci, Stefano; Butts, Craig P.; Bifulco, Giuseppe | |
| Identification and mechanism of action analysis of the new PARP-1 inhibitor 2″-hydroxygenkwanol A | 1-gen-2015 | Dal Piaz, Fabrizio; Ferro, Piera; Vassallo, Antonio; Vasaturo, Michele; Forte, Giovanni; Chini, Maria Giovanna; Bifulco, Giuseppe; Tosco, Alessandra; De Tommasi, Nunziatina | |
| Natural iminosugar (+)-lentiginosine inhibits ATPase and chaperone activity of Hsp90 | 1-gen-2012 | Dal Piaz, Fabrizio; Vassallo, Antonio; Chini, Maria Giovanna; Cordero Franca, M.; Cardona, Francesca; Pisano, Claudio; Bifulco, Giuseppe; De Tommasi, Nunziatina; Brandi, Alberto | |
| Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells | 1-gen-2018 | Khalfaoui, Ayoub; Chini, Maria G.; Bouheroum, Mohamed; Belaabed, Soumia; Lauro, Gianluigi; Terracciano, Stefania; Carmela Vaccaro, Maria; Bruno, Ines; Benayache, Samir; Mancini, Ines; Bifulco, Giuseppe | |
| Molecular mechanism of tanshinone IIA and cryptotanshinone in platelet anti-aggregating effects: an integrated study of pharmacology and computational analysis | 1-gen-2015 | Maione, Francesco; Cantone, Vincenza; Chini, MARIA GIOVANNA; DE FEO, Vincenzo; Mascolo, Nicola; Bifulco, Giuseppe | |
| Structure-Based Discovery of Inhibitors of Microsomal Prostaglandin E2 Synthase-1, 5-Lipoxygenase and 5-Lipoxygenase-Activating Protein: Promising Hits for the Development of New Anti-inflammatory Agents | 1-gen-2011 | De Simone, R.; Chini, M. G.; Bruno, I.; Riccio, R.; Mueller, D.; Werz, O.; Bifulco, G. | |
| Fusicoccane Diterpenes from Hypoestes forsskaolii as Heat Shock Protein 90 (Hsp90) Modulators | 1-gen-2019 | D'Ambola, Massimiliano; Fiengo, Lorenzo; Chini, Maria Giovanna; Cotugno, Roberta; Bader, Ammar; Bifulco, Giuseppe; Braca, Alessandra; De Tommasi, Nunziatina; Dal Piaz, Fabrizio | |
| Discovery of new molecular entities able to strongly interfere with Hsp90 C-terminal domain | 1-gen-2018 | Terracciano, Stefania; Russo, Alessandra; Chini, Maria G.; Vaccaro, Maria C.; Potenza, Marianna; Vassallo, Antonio; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| The bile acid receptor GPBAR-1 (TGR5) modulates integrity of intestinal barrier and immune response to experimental Colitis | 1-gen-2011 | Cipriani, S.; Mencarelli, A.; Chini, M. G.; Distrutti, E.; Renga, B.; Bifulco, G.; Baldelli, F.; Donini, A.; Fiorucci, S. | |
| Elucidating new structural features of the triazole scaffold for the development of mPGES-1 inhibitors | 1-gen-2015 | Chini, MARIA GIOVANNA; Ferroni, Claudia; Cantone, Vincenza; Dambruoso, Paolo; Varchi, Greta; Pepe, Antonella; Fischer, Katrin; Pergola, Carlo; Werz, Oliver; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe | |
| Computational NMR Methods in the Stereochemical Analysis of Organic Compounds: Are Proton or Carbon NMR Chemical Shift Data More Discriminating? | 1-gen-2015 | Chini, MARIA GIOVANNA; Riccio, Raffaele; Bifulco, Giuseppe | |
| Structural basis for the design and synthesis of selective HDAC inhibitors | 1-gen-2013 | DI MICCO, Simone; Chini, MARIA GIOVANNA; Terracciano, Stefania; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe | |
| Discovery That Theonellasterol a Marine Sponge Sterol Is a Highly Selective FXR Antagonist That Protects against Liver Injury in Cholestasis | 1-gen-2012 | Barbara, Renga; Andrea, Mencarelli; Claudio, D'Amore; Sabrina, Cipriani; Maria Valeria, D'Auria; Valentina, Sepe; Chini, MARIA GIOVANNA; Monti, Maria Chiara; Bifulco, Giuseppe; Angela, Zampella; Stefano, Fiorucci | |
| Design and synthesis of a second series of triazole-based compounds as potent dual mPGES-1 and 5-lipoxygenase inhibitors | 1-gen-2012 | Chini, Maria Giovanna; De Simone, Rosa; Bruno, Ines; Riccio, Raffaele; Dehm, Friederike; Weinigel, Christina; Barz, Dagmar; Werz, Oliver; Bifulco, Giuseppe | |
| A Novel Potent Nicotinamide Phosphoribosyltransferase Inhibitor Synthesized via Click Chemistry | 1-gen-2010 | G., Colombano; C., Travelli; U., Galli; A., Caldarelli; Chini, MARIA GIOVANNA; P. L., Canonico; G., Sorba; Bifulco, Giuseppe; G. C., Tron; A. A., Genazzani |
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