CHINI, Maria Giovanna

CHINI, Maria Giovanna  

DIPARTIMENTO DI BIOSCIENZE E TERRITORIO  

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Risultati 1 - 20 di 76 (tempo di esecuzione: 0.031 secondi).
Titolo Data di pubblicazione Autore(i) File
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines 1-gen-2023 De Vita, Simona; Meninno, Sara; Capasso, Lucia; Colarusso, Ester; Chini, Maria Giovanna; Lauro, Gianluigi; Rinaldi, Romolo; De Cicco, Annalisa; Sian, Veronica; Terracciano, Stefania; Nebbioso, Angela; Lattanzi, Alessandra; Bifulco, Giuseppe
4-Methylenesterols from Theonella swinhoei sponge are natural pregnane-X-receptor agonists and farnesoid-X-receptor antagonists that modulate innate immunity 1-gen-2012 De Marino, Simona; Ummarino, Raffaella; Valeria D’Auria, Maria; Chini, Maria Giovanna; Bifulco, Giuseppe; D’Amore, Claudio; Renga, Barbara; Mencarelli, Andrea; Petek, Sylvain; Fiorucci, Stefano; Zampella, Angela
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis 1-gen-2022 Colarusso, E; Gazzillo, E; Boccia, E; Giordano, A; Chini, Mg; Bifulco, G; Lauro, G
A Chemical-Biological Study Reveals C-9-type Iridoids as Novel Heat Shock Protein 90 (Hsp90) Inhibitors 1-gen-2013 Dal Piaz, F.; Vassallo, A.; Temraz, A.; Cotugno, R.; Belisario, M. A .; Bifulco, G.; Chini, M. G.; Pisano, C.; De Tommasi, N.; Braca, A.
A Novel Potent Nicotinamide Phosphoribosyltransferase Inhibitor Synthesized via Click Chemistry 1-gen-2010 G., Colombano; C., Travelli; U., Galli; A., Caldarelli; Chini, MARIA GIOVANNA; P. L., Canonico; G., Sorba; Bifulco, Giuseppe; G. C., Tron; A. A., Genazzani
Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19) 1-gen-2020 De Vita, S.; Chini, M. G.; Lauro, G.; Bifulco, G.
Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches 1-gen-2021 Chini, M. G.; Lauro, G.; Bifulco, G.
Anti-inflammatory and analgesic activity of carnosol and carnosic acid in vivo and in vitro and in silico analysis of their target interactions 1-gen-2017 Maione, Francesco; Cantone, Vincenza; Pace, Simona; Chini, Maria Giovanna; Bisio, Angela; Romussi, Giovanni; Pieretti, Stefano; Werz, Oliver; Koeberle, Andreas; Mascolo, Nicola; Bifulco, Giuseppe
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests 1-gen-2021 De Vita, Simona; Chini, Maria Giovanna; Saviano, Gabriella; Finamore, Claudia; Festa, Carmen; Lauro, Gianluigi; De Marino, Simona; Russo, Roberto; Avagliano, Carmen; Casapullo, Agostino; Calignano, Antonio; Bifulco, Giuseppe; Iorizzi, Maria
Can Small Chemical Modifications of Natural Pan-inhibitors Modulate the Biological Selectivity? the Case of Curcumin Prenylated Derivatives Acting as HDAC or mPGES-1 Inhibitors 1-gen-2015 Iranshahi, Mehrdad; Chini, MARIA GIOVANNA; Masullo, Milena; Sahebkar, Amirhossein; Javidnia, Azita; Chitsazian Yazdi, Mahsa; Pergola, Carlo; Koeberle, Andreas; Werz, Oliver; Pizza, Cosimo; Terracciano, Stefania; Piacente, Sonia; Bifulco, Giuseppe
Carnosol Attenuates LPS-Induced Inflammation of Cardiomyoblasts by Inhibiting NF-κB: A Mechanistic in Vitro and in Silico Study 1-gen-2022 Baradaran Rahimi, Vafa; Momeni-Moghaddam, Mohammad Amin; Chini, Maria Giovanna; Saviano, Anella; Maione, Francesco; Bifulco, Giuseppe; Rahmanian-Devin, Pouria; Jebalbarezy, Ali; Askari, Vahid Reza
Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A 1-gen-2024 Capuano, Alessandra; D’Urso, Gilda; Aliberti, Michela; Ruggiero, Dafne; Terracciano, Stefania; Festa, Carmen; Tosco, Alessandra; Chini, Maria Giovanna; Lauro, Gianluigi; Bifulco, Giuseppe; Casapullo, Agostino
Computational NMR Methods in the Stereochemical Analysis of Organic Compounds: Are Proton or Carbon NMR Chemical Shift Data More Discriminating? 1-gen-2015 Chini, MARIA GIOVANNA; Riccio, Raffaele; Bifulco, Giuseppe
Conformationally locked calixarene-based histone deacetylase inhibitors 1-gen-2010 Chini, M. G.; Terracciano, S.; Riccio, R.; Bifulco, G.; Ciao, R.; Gaeta, C.; Troisi, F.; Neri, P.
Conicasterol E, a Small Heterodimer Partner Sparing Farnesoid X Receptor Modulator Endowed with a Pregnane X Receptor Agonistic Activity, from the Marine SpongeTheonella swinhoei 1-gen-2012 Sepe, Valentina; Ummarino, Raffaella; Valeria D’Auria, Maria; Chini, Maria Giovanna; Bifulco, Giuseppe; Renga, Barbara; D’Amore, Claudio; Debitus, Cécile; Fiorucci, Stefano; Zampella, Angela
Correction: Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors 1-gen-2016 Terracciano, Stefania; Chini, Maria Giovanna; Vaccaro, Mariacarmela; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Cytotoxic Sesquiterpenoids from Ammoides atlantica Aerial Parts 1-gen-2021 Boudermine, S.; Parisi, V.; Lemoui, R.; Boudiar, T.; Chini, M. G.; Franceschelli, S.; Pecoraro, M.; Pascale, M.; Bifulco, G.; Braca, A.; De Tommasi, N.; De Leo, M.
Design and synthesis of a second series of triazole-based compounds as potent dual mPGES-1 and 5-lipoxygenase inhibitors 1-gen-2012 Chini, Maria Giovanna; De Simone, Rosa; Bruno, Ines; Riccio, Raffaele; Dehm, Friederike; Weinigel, Christina; Barz, Dagmar; Werz, Oliver; Bifulco, Giuseppe
Design, Synthesis, and Biological Activity of Hydroxamic Tertiary Amines as Histone Deacetylase Inhibitors 1-gen-2012 Terracciano, Stefania; Chini, Maria Giovanna; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
DFT/NMR integrated approach: a valid support to the total synthesis of chiral molecules 1-gen-2008 Chini, M. G.; Riccio, R; Bifulco, G